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| Hans-Günter Meyer-Thompson | Naloxon

Fentanyl-Type Antagonist of the μ-Opioid Receptor: Important Role of Axial Chirality in the Active Conformation. 

Fentanyl-Type Antagonist of the μ-Opioid Receptor: Important Role of Axial Chirality in the Active Conformation. 

Arita H, Tanaka R, Kikukawa S, Tomizawa T, Sakata H, Funada M, Tomiyama K, Hashimoto M, Tasaka T, Tabata H, Nakamura K, Makino K, Oshitari T, Natsugari H, Takahashi H. 

J Med Chem. 2024 Jun 27;67(12):10447-10463. doi: 10.1021/acs.jmedchem.4c00935. Epub 2024 Jun 13. PMID: 38869493; PMCID: PMC11215721.

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11215721/